Thanzi, Kukonzekera
"Olanzapine": analogues, malongosoledwe mankhwala, malangizo ntchito
Zochizira oyambitsa misala ndi ochititsa kuti matenda ntchito mankhwala pamaziko a mankhwala olanzapine. Pali mankhwala ambiri ndi mayina osiyanasiyana malonda, koma yemweyo antipsychotic kwenikweni. Mmodzi mankhwala oterewa ndi mankhwala "olanzapine" analogs ali mu kapangidwe kake okwana yogwira pophika.
Kufotokozera lokonzekera
Izi zachitika mwa nthumwi antipsychotic "ALSI Pharma" ZAO monga kuwala mapiritsi chikasu, mawonekedwe a omwe akufanana ndi yamphamvu biconvex.
Kapangidwe ka mankhwala kupanga zosakaniza wofooka, monga microcrystalline mapadi mtundu, lactose monohydrate, krospovidonovy filler, magnesium stearate. chiwerengero chawo chinawonjezeka mu nthawi ziwiri, zitatu kapena zinayi, malinga ndi mlingo olanzapinovoy.
magome ali odzaza Mlingo onse zidutswa 7 matuza mu paketi zimenezi 4 kapena 8 zidutswa.
Amatanthauza "olanzapine" wogwiritsa Phunziro pankhaniyi zikugwirizanirana ndi mankhwala antipsychotic neuroleptic amene kuonetsa kuyandikana kwa serotonin, dopamine, muscarinic, adrenergic ndi histamine cholandilira mapangidwe.
Kusankha yafupika ntchito excitatory wa mesolimbic manyuroni dopaminergic, kugwira ntchito pang'ono mu striatal mitsempha conduction, amene nthawi machitidwe a injini. Utachepa mphamvu mu bongo ochiritsira zoteteza, ngati inu ntchito mlingo wochepa popanda kuchititsa cataleptic tulo.
Medicine "Olanzapine" kumawonjezera anxiolytic efficacy mayeso ntchito "anxiolytic" pamene anali akuthamanga. Akuchita mavuto obwera ndi zoipa zipatso monga zinyengo ndi masomphenya hallucinatory.
Kodi ntchito
Miyala "olanzapine" zotsatira amagwiritsa ntchito pa boma schizophrenic mu akula mu gawo pachimake, ngati posungira ndi yaitali protivopovtornogo chithandizo. Iwo amagwiritsa ntchito matenda psychotic ndi zizindikiro kuberekana kwa zinyengo, masomphenya hallucinatory ndi zizindikiro zoipa monga flattening maganizo, kuchepetsa ntchito chikhalidwe kwambiri, zikutha m'mayiko zida ntchito mawu.
Mankhwala inathetsedwa zisadzachitikenso a khunyu ndi matenda osokonezeka maganizo, ngati phale bwinobwino kuchitira magawo wosangalala monyanyira.
Kukonzekera "olanzapine" inakhazikitsa akulu ndi matenda ochititsa kuti affective mu mawonekedwe a monotherapy kapena molumikizana ndi medicaments munali lifiyamu ayoni kapena asidi valproic. mankhwala amagwiritsidwa ntchito pofuna kuchiza pachimake wosangalala monyanyira kapena wosanganiza mitundu ya zinthu zimene zingachitike mbali psychotic, komanso ndi kusala kusintha pang'onopang'ono.
Kumatanthauza pamodzi ndi mankhwala fluoxetine zinthu kuvutika kuti imakhudzana ndi matenda osokonezeka maganizo.
Terms of ntchito
Medicine "olanzapine" wogwiritsa ntchito malangizo tsiku 0,005 kuti 0,02 ga pakamwa popanda kum'mamatira mphamvu mode.
boma schizophrenic odwala wamkulu mankhwala koyamba tsiku mlingo wa 0,010 ga
Wamkulu pachimake kukonda, ochititsa kuti matenda yodziwika ndi, kuchotsedwa kuchuluka tsiku la olanzapine mu 0.015 ga, amene kutumikiridwa kamodzi. Ngati miyala ntchito posungira zotsatira molumikizana ndi mankhwala zochokera lifiyamu ion kapena asidi valproic, ndiye kutumikiridwa mu mlingo tsiku la 0,010 ga pa kamodzi.
njira kuvutika mu akula chifukwa matendaŵa, kuthetsa kuchuluka tsiku la 0,005 ga, ndi pamodzi 0,020 ga fluoksetinovogo mankhwala. Ngati pali kufunika, ndiye amaloledwa kusintha kwa dosing wa mankhwala.
Kwa odwala achikulire zotheka aakulu kuopseza insufficiency aimpso kapena chiwindi aakulu monga pamene pali mavuto kugwirizana ndi jenda wamkazi, senile zaka pamene deceleration kuwombola olanzapine tsiku koyamba kuchuluka yafupika 0,005 ga
zida
Medicament "Olanzapine" Akhristu ali maina malonda osiyana. Iwo amapangidwa ndi opanga zoweta ndi achilendo.
Pakati pa opanga Russian wa sapota-kuchokera makampani 'mankhwala matekinoloje "ndi mankhwala" Olanzapine-TL ", mu mawonekedwe piritsi 0,0025 ga filimu TACHIMATA.
mankhwala ena m'banja njira "Olanzapine" chopangidwa ndi JSC "North Star". Pali piritsi ndi ❖ kuyanika filimu ndi mlingo wa 0,005 ga
Russian fakitale "Kanonfarma Yopanga" JSC umatulutsa mankhwala "Canon of olanzapine."
mankhwala Israel ndi mankhwala "Olanzapine Teva," makampani kupanga "Teva mankhwala ogwira Co., Ltd.".
Chisiloveniya analogue ndi amatanthauza "Zalasta Cu tsamba", mapiritsi a 0,015 ga wopita resorption. Anapanga ndi ogwira "Krka, Novo mesto." Komanso deta umatulutsa mankhwala "Zalasta" miyala.
Swiss analogue mankhwala imatengedwa "Zyprexa" monga lyophilisate mu mbale, amene njira okonzekera makonzedwe mu mnofu, ndi mlingo wa 0,010 mu dispersible piritsi mawonekedwe 0.005 magalamu alipo mankhwala "Zyprexa Zidis". Iwo amapangidwa ndi "Eli Lilly Vostok SA". Mu msika mankhwala pali "Zyprexa Adair" ufa medicament choperekedwa 0,21 ga
Polish kampani ya "Polpharma" mankhwala chopangidwa "Normiton" miyala ndi m'chimake ❖ kuyanika wa 0.005 ga
Mankhwala "Olanzapine" Chihangare Anzawo ndi "Gidiyoni Richter" otchedwa mapiritsi "Parnasan" ndi mankhwala chomera "EGIS" anayamba mankhwala "Egolanza".
Kufotokozera "Zalasta" mankhwala
Izi amatanthauza neuroleptic antipsychotic. Kuwala mapiritsi achikasu ozungulira, pang'ono biconvex mawonekedwe ndi yamawangamawanga mdima. Pali Mlingo asanu: 0,0025 G 0,005 ga, 0.01 ga, 0,015 ga ndi 0,02 ga olanzapine. zigawo zina ankaona anafooka Cellactose, wowuma pregelatinized ndi chimanga mawonekedwe, kuliumitsa aerosilovy pophika, magnesium stearate.
Imasonyeza piritsi mawonekedwe "Zalasta" malangizo Buku limafotokoza kalembedwe mu mawonekedwe a zojambula mochita kugoba ndi kumasonyeza mlingo. Kugula katundu ndi contoured mbale mapiritsi 7. paketiyo anyamula 4 kapena 8 matuza amenewa.
Izi wothandizila neuroleptic akusonyeza ntchito yotakata pharmacological. Antipsychotic zotsatira kugwirizana ndi mtundu interlock formations dopamine cholandilira. ntchito Sedative chifukwa braking malo adrenoceptor zomwe zimapanga ndi reticular mapangidwe ku maselo a tsinde ubongo.
ntchito Antiemetic n'zotheka pa amasiya D 2 cholandilira -dopaminovogo gawo mu choyambitsa-mtundu zone limene lili pakati emetic.
udindo Hypothermic ikuchitika ndi kutsekereza dopamine cholandilira formations mitundu mu ubongo imene imalamulira kutentha kwa.
Medicine "Zalasta" malangizo Buku zikusonyeza ntchito pa mawonetseredwe schizophrenic. Mapiritsi ali wokhoza kusunga mwachangu kusintha zizindikiro matenda pa nthawi yaitali mankhwala a odwala ndi zotsatira koyamba zabwino mankhwala.
Amatanthauza kuthetsa episodic kukonda pakati kapena zovuta mawonekedwe. Mapiritsi makhalidwe kuchenjeza mpheto kubwerezabwereza akamakonda matendaŵa anthu ndi nkhani wosangalala monyanyira.
mankhwala cholinga cha utsogoleli m'kamwa kamodzi pa tsiku. particles chakudya sikungawononge mayamwidwe ndondomeko ya olanzapine, zomwe zimathandiza kuti ntchito piritsi nthawi iliyonse. Pa Kulipira mankhwala ayenera pang'onopang'ono kuchepetsa mlingo.
Zochizira matenda schizophrenic ntchito dosing koyamba magalamu 0,010 patsiku.
Magawo a kukonda amayamba ankachitira mlingo tsiku la 0.015 ga, amene kutumikiridwa mu ntchito limodzi kapena magalamu 0,010 pamene pamodzi neuroleptics ena.
kupewa kubwereza kwa matendaŵa ku attenuation sitepe ikuchitika yaikulu yopereka medicament magalamu 0,010 patsiku. Ngati anthu kutenga chida pothetsa episodic kukonda, kuti likhale mankhwala ntchito mlingo chomwecho. M'pofunika kuonjezera kuchuluka kwa mankhwala mwambo episodic mawonetseredwe latsopano kapena m'magulu maganizo komanso kuwonjezera mankhwala a disruptions maganizo.
Mlingo tsiku la medicament kuthetsa matenda schizophrenic, nkhani wosangalala monyanyira ndi matenda ochititsa kuti kuchenjeza akubwereza ntchito ku 0,005 kuti 0,020 ga Mtengo wa potsata magawo matenda a wodwalayo.
Okalamba m'munsi koyamba mlingo wa ku 0.005 ga si analangiza Koma zimenezi idzagwira ntchito kwa Odwala ndi zaka 65, ngati pali mfundo zoopsa.
Kufotokozera "Olanzapine Canon" mankhwala
Zimenezi wa neuroleptic antipsychotic medicament ndi alembedwe piritsi TACHIMATA ndi m'chimake a. The mawonekedwe miyala yochititsa ndi pamalo awiri otukukira kunja chikasu, zili mkati mwa mtundu womwewo.
Lilili mu Mlingo awiri: pa 0,005 ga ndi 0.01 ga olanzapine. The zosakaniza wothandiza monga hydroxypropyl mapadi ndi M'MALO otsika, calcium mankwala a hydrogen, croscarmellose sodium, mannitol, magnesium stearate.
M'chimake chikasu Opadry filimu aumbike mwa mtundu wachiwiri, polyvinyl mowa, macrogol, talc, titaniyamu dioxide, chitsulo okusayidi.
mankhwala analamula kuti impairments, chifukwa chochititsa ndi kugwiritsa yaitali antirelapse odwala wamkulu akudwala matenda schizophrenic.
mankhwalawo ikuchitika monotherapy ndi osakaniza mayikidwe ndi lifiyamu pawiri ndi mtundu wamphamvu nkhani wosangalala monyanyira kapena wosanganiza wa ochititsa kuti affective matenda, ndiwo mawu ndi psychotic ndi kudya kusintha mbali. Mankhwala ochiza matendawa kubwereza anthu ndi matenda osokonezeka maganizo, ngati mankhwala athandizikira ndi gawo wosangalala monyanyira.
Mankhwalawa akulu ndi maganizo chifukwa cha matendaŵa, komanso khola digiri maganizo mankhwala "Canon Olanzapine", ndi neuroleptic, akhoza pamodzi ndi wothandizila munali fluoxetine.
Amatengedwa pakamwa, osati chotsatira chakudya. Guide akuonetsa kuti mlingo akangofika medicament, ndilo tsiku, chiwerengero cha 0,005-0,020 njira amasankhidwa payekha kwa wodwala aliyense malingana ndi zizindikiro matenda.
matenda Schizophrenic wamkulu mtima kuchitira koyamba tsiku dosing mankhwala mu 0.010 ga, amene kutumikiridwa mwakamodzi.
Ulili ochititsa kuti matenda pachimake kukonda kuthetsa mlingo tsiku la mankhwala kwa 0,015 ga kapena 0,010 ga olanzapine pamodzi ndi wothandizila munali lifiyamu ayoni kapena asidi valproic.
Zikuthandiza ntchito matendaŵa pa koyamba dosing tsiku ikuchitika odwala 0.010 chitachitidwa ngati phwando la medicament chifukwa kukonda pachimake, tiyenera kugwiritsa ntchito zinthu mu mulingo womwewo.
matenda a maganizo kugwirizana ndi matenda matenda odwala wamkulu mankhwala osakaniza 0,005 ga ndi 0,020 ga kukonzekera olanzapine fluoksetinovyh amene kutumikiridwa madzulo.
Antidepressive zotsatira za mankhwala akuwonetseredwa mu ndalama kuchokera magalamu 0,006 kuti 0,012 ndi avareji dosing tsiku ndi tsiku 0,0074 ga mlingo mankhwala fluoksetinovyh ranges kuchokera 0,025 kuti 0,030 ga Ngati pali kufunika, n'zotheka abwereze ndi dosing wa mankhwala onse.
Achire khola mawonekedwe maganizo chikutha ndi osakaniza 0,005 ga ndi 0,02 ga njira olanzapine fluoksetinovyh amene kutumikiridwa kamodzi madzulo.
Kufotokozera "Zyprexa" mankhwala
neuroleptic iyi inatulutsa mu mawonekedwe piritsi TACHIMATA ndi m'chimake a. Pali zinthu zinayi mlingo chiphunzitso: 0,0025 pa 0,005, 0,010 ndi 0,0075 kwa ×, Y zomwe ndi zoyenerera kalembedwe padziko «Lilly 4112», «Lilly 4115», «Lilly 4116», «Lilly 4117".
zosakaniza amangokhala mu mawonekedwe a lactose, hydroxypropylcellulose, crospovidone, microcrystalline mapadi mtundu dongosolo aumbike mankhwala mankhwala enaake a stearate.
mapiritsi ndi mmatumba mu matuza zidutswa 7 paketi lili 4 mizere ma CD.
Palinso amaundana-zouma mawonekedwe, anafuna kupanga njira mu mnofu. Yellow madzi mlingo 0.01g mmatumba mu mbale. zigawo amangokhala amaonedwa lactose monohydrate acid tartaric.
Mankhwala akusonyeza zotsatira antipsychotic.
The yogwira pophika medicament ndi khalidwe ngati ligand chimango ndi serotonin, dopamine, mamita-choline, H1-histamine ndi alpha1-cholandilira formations adrenozavisimymi. Olanzapine kumakhudza kusankha pa boma la dongosolo limbic.
Mankhwala "Zyprexa" malangizo ntchito limalangiza kugwiritsa ntchito bwino za khwerero amphamvu matenda schizophrenic ndi psychotic amene anatsagana ndi zizindikiro bwino zinyengo, kuyerekezera zinthu m'maganizo, matenda ganizo, ovuta maganizo Muzisamala kapena mtundu zoipa mu mawonekedwe a maganizo ndi chikhalidwe chowasiyanitsa, matenda a zida ntchito mawu. mankhwala lasonyezedwa kwa kuchotsa zizindikiro sekondale affective chifukwa cha matenda schizophrenic.
Piritsi "Zyprexa" malangizo Buku amalimbikitsa kumwa pakamwa, nthawi iliyonse. mankhwala oyambirira a mlingo umodzi ndi 0,010 ga Kenako mlingo tsiku ranges kuchokera 0,005 kuti 0,020 ga, amene ananamizira ndi symptomatic chithunzi.
Intramuscularly jekeseni mankhwala ngati pakufunika kuti asiye ndi malemeredwe psychomotor khalidwe anthu ndi oyambitsa misala, matenda ochititsa kuti affective ndi maganizo.
Pamaso ntchito, lyophilisate anali sitimadzipereka mu 2.1 ml ya jekeseni amadzimadzi sing'anga. A njira bwino ndi kum'chitira chikasu.
Chisangalalo mantha wachisokonezo schizophrenic ndi ochititsa kuti avule mmodzi-mlingo wa 0,010
Poganizira tsopano wodwalayo achire mobwerezabwereza ka mlingo 0,010 ga anachita pambuyo Mph 120 kuchokera ntchito loyamba ndi awa 0,010 ga ankadya pambuyo Mphindi 240 kuchokera kudzolanso.
Pakuti zina mankhwala "Zyprexa" kusuntha kwa mawonekedwe ake piritsi ndi mlingo wa ku 0,005 kuti 0,020 ga
Kusakhazikika mu maganizo kuchotsedwa mu umodzi mlingo mu mnofu wa 0,0025 Poona chithunzi matenda a mtima, wachiwiri makonzedwe mlingo 0.005g ikuchitika pambuyo Mphindi 120 kuchokera ntchito choyamba.
Mankhwala akuti "Adair Zyprexa"
Pali medicament "olanzapine" analogs kuti amapangidwa mu mawonekedwe ufa ndi 0,405 ga olanzapine mu mbale ndi syringe zosungunulira ndi singano.
Amatanthauza "Adair Zyprexa" amatanthauza antipsychotic neuroleptic mankhwala ntchito.
Mankhwala limaleka kuwonongeka, ntchito kwa posungira ndi yaitali mankhwala a protivopovtornogo schizophrenic ndi kusintha maganizo ndi zizindikiro za mkulu-zokolola mu mawonekedwe a zinyengo, masomphenya hallucinatory ndi zoipa maganizo flattening, zatha ndi zida amapilira.
Mankhwala kuchitira aakulu wosangalala monyanyira ndi ophatikizana nkhani ya matendaŵa, imene n'zotheka mbali psychotic ndi kusintha mwamsanga pang'onopang'ono.
Koyamba tsiku mlingo ntchito ndi 0.010 kapena 0.015, tsiku kuchuluka kwa mankhwala akanasankhidwa wodwala aliyense payekha, kutenga nkhani chithunzi matenda. Amagwiritsidwa ntchito mlingo achire tsiku la ku 0,005 kuti 0,020 ga
Kuwonjezeka mlingo zimatheka ndi zotsatira za kafukufuku. Kuwonjezeka kuchuluka kwa mankhwala ikuchitika mu masiteji, tsiku lililonse.
odwala achikulire koyamba tsiku mlingo mu kukhalapo kwa impso ntchito osakwanira ndi chiwindi tisonyezeni 0.005 ga
mtengo analogues
assortment Large wa antipsychotics limakupatsani kusankha mankhwala woyenera, womwe abwino khalidwe ndi mtengo. Mankhwala "Olanzapine" mtengo wochepa. Kenaka miyala zikhoza kugulidwa kwa 290 rubles.
Mankhwala "Zalasta" mtengo kuchokera 1370 rubles.
Mtengo njira ankaona mapiritsi "Zidis Zyprexa." Kuti phukusi mankhwala ayenera kulipira 2370 rubles. Mtengo analogi wa "Ku-Tab Zalasta" ndi 1075 rubles.
Pa mankhwala "Zyprexa" mtengo filimuyo negative. Paketi mapiritsi 28 ndalama 4760 rubles.
Magulu ovutika lidzakhala lilipo mankhwala "Olanzapine" imene ili nusu ya mtengo.
Views odwala
Za mankhwala "Olanzapine" ndemanga angamvele zabwino ndi zoipa. mankhwala ambiri amathandiza maganizo ndi kuchepetsa maganizo patapita masiku ochepa mankhwala. Iye ndi chimodzi cha mphamvu ya neuroleptics, amene Amachepetsa wodwala, kumatha nkhawa.
Mwa kuipa kwa zimatulutsa zotsatira osafunika amene anagwirizana ndi liwiro la kagayidwe, chifukwa kuchuluka thupi la wodwalayo. Somnolence, asthenia syndrome, chizungulire, magazi orthostatic akhoza kusiya mtundu kuthamanga kukhala minofu zofewa kutupa ndi dryness wa nembanemba mucous.
Kwa ena odwala, ngakhale mlingo ka mankhwala ndi sedative amphamvu, kumene kugona kwa maola 12 pa tsiku.
Thupi osiyana Komabe, ndi miyala zinthu zosiyana kwa wodwala aliyense. Pakuti kusankha njira zomwe ndi zoyenerera kufunsa dokotala.
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