Thanzi, Kukonzekera
"Lomfloks": malangizo ntchito, mtengo, analogs
N'chifukwa mankhwala monga "Lomfloks" awerenge? Malangizo ntchito, contraindications ndi zizindikiro yolandirira mankhwala Adzaperekedwa mwatsatanetsatane m'nkhani ino. Komanso, kwa izo mudzaphunzira za mankhwala alipo, amene zinthu gawo la ilo, momwe ndalama ndi ngati iye analogs mtundu uliwonse.
Kenaka mankhwala, mawonekedwe ake, kufotokoza ndi zikuchokera
Mu mawonekedwe ndi zimene mankhwala chikupezeka monga "Lomfloks"? Malangizo ntchito kudziŵitsa kuti medicament yogwira ndi akugulitsa kokha mu mawonekedwe a mapiritsi lokutidwa (filimu) oblong miyala (400 mg) monga kuwala bulauni mtundu.
The yogwira zikuluzikulu za wothandizila izi lomefloxacin (ntchito ngati hydrochloride a). Pankhani zigawo zina, ndiye iwo monga lactose, woyeretsedwa talc, wowuma, crospovidone, polyvinylpyrrolidone, sodium lauryl sulphate propylene glycol, mankhwala enaake a stearate, ndi sodium wowuma glycolate ndi colloidal pakachitsulo woipa.
The zikuchokera chipolopolo atsatire zinthu: methylene enaake, isopropanol, titaniyamu woipa ndi hydroxypropyl methylcellulose.
"Lomfloks" ndi miyala iwiriyo matuza (5 zidutswa) anayikidwa mu makatoni.
Monga ntchito mankhwala?
ndi mankhwala "Lomfloks" n'chiyani? Malangizo ntchito zikusonyeza kuti wothandizila izi ndi kupanga antimicrobial wothandizira. Adzaupereka kwa gulu fluoroquinolone mankhwala ndipo ali ndi sipekitiramu lonse kanthu bactericidal.
Akuti mankhwala angathe kutsekereza mabakiteriya DNA gyrase, potero kupanga tetramer ndi zovuta zake ndi kusokoneza kugawanika ndi galamafoniyo ya DNA. Chifukwa cha kukhudzana ngati pali kuwonongedwa kwa maselo tizilombo.
medicament Ichi ndi yogwira motsutsana galamu zoipa ndipo ndi galamu tizilombo zabwino ndi aerobes. Komanso, mankhwala zimawononga zimakhudzanso mauka, Mycobacterium TB (intra- ndi extracellularly ili), komanso ena tizilombo ta uroplazmy ndi mycoplasma.
M'madera acidic efficacy mankhwala ali kwambiri yafupika, ndi kukana akufotokozera pang'onopang'ono.
Mankhwala ali ndi kutchulidwa zotsatira postantibioticski.
Tiyenera kuona kuti streptococci ndi anaerobes ndi kugonjetsedwa ndi zochita za lomefloxacin.
Pharmacokinetics
liti mankhwala odzipereka "Lomfloks" (mapiritsi)? Ogwiritsa ntchito limanena kuti pambuyo makonzedwe mu chigawo ake yogwira pafupifupi atamezedwa kotheratu kwa mundawo m'mimba.
Pogwiritsa 400 mg wa chiphunzitso ndende ake apamwamba mu magazi anaona pambuyo maola 1.5-2 ndipo watsala 3,2-5,2 mg wa pa lita. Tiyeneranso kukumbukira kuti pamene kulandira medicament mu anati mlingo lomefloxacin woipa akhoza kupitiliza MIKA kuti mabakiteriya ambiri. Osachepera theka tsiku.
Communication yogwira mankhwala kwa mapulotini plasma pafupifupi 10%. Lomefloksatsin mwachilungamo mwamsanga likulowerera mu zimakhala zonse za thupi. The ndende ya mankhwala mu madzi enieni nthawi 3-6 kuposa mu plasma, makamaka Prostate zimakhala, macrophages m'mapapo ndi mkodzo.
The theka moyo wa chinthu yogwira pafupifupi 7-9 maola. Pafupifupi 70-80% ya lomefloxacin ndi linanena bungwe masana (mu mawonekedwe unmodified) mu mkodzo.
Odwala ndi mkhutu impso ntchito theka moyo wa chinthu yogwira ali kwambiri.
umboni
Amene matenda prescribers "Lomfloks"? Malangizo ntchito lili ndi zizindikiro zotsatirazi:
- matenda kupuma (matenda), kapena kani, magulu awo m'munsi (kuphatikizapo exacerbation wa chifuwa ndi chibayo);
- matenda opatsirana ndi yotupa kuti akhala ndi bakiteriya tcheru lomefloxacin;
- otitis TV;
- aakulu ndi pachimake chlamydial, gonococcal matenda, kuphatikizapo;
- Matenda ovuta wopepuka wa mkodzo ndi machitidwe ubereki;
- matenda opatsirana a zimakhala zofewa ndi khungu;
- cholecystitis ndi enterocolitis opatsirana;
- matenda zimfundo ndi mafupa, kuphatikizapo osteomyelitis aakulu;
- TB m'mapapo mwanga (kuphatikizapo mitundu pachimake pang'onopang'ono kwa matenda, mankhwala kusamva mabakiteriya, tsankho rifampicin, concomitant TB nonspecific yotupa njira).
Komanso dziwani kuti mankhwala ankaona zambiri analamula kuti kupewa mavuto opatsirana njira opaleshoni transurethral.
contraindications
Ngati pali kuvutika Mulimonsemo sangathe kutenga miyala "Lomfloks"? Malangizo ntchito (mtengo wa mankhwala ali anatchula pansipa) lili mndandanda wa contraindications:
- pa gestation ndi yoyamwitsa;
- khunyu, arteriosclerosis oziziritsa, komanso boma, limodzi ndi khunyu;
- Ana kwa zaka 15;
- mtima hypersensitivity kuti lomefloxacin ndi quinolones ena.
Medicament "Lomfloks": malangizo ntchito
Kufotokozera za chida ichi nthawi zonse zilipo malangizo Ufumuyo. Komanso, Zamkati kuti mankhwala kudziŵitsa odwala zimene kumwa mankhwala ayenera kumwedwa pa kupatuka anapatsidwa.
Miyala "Lomfloks" ayenera ingest (chakumwa madzi firiji). nchito zake sikudalira kudya chakudya. Mlingo watsiku ndi chiphunzitso ichi ndi 400 mg tsiku lililonse.
Pamene chakhungu impso ntchito mu tsiku loyamba la mankhwala Kwalamulidwa 400 mg wa mankhwala, ndi lotsatira - 200 mg (kamodzi pa tsiku). Mlingo ndi nthawi ya mankhwala zimadalira kuopsa kwa kupatuka alipo ndi chiwopsezo.
Kukachitika kuti wodwala matenda ndi mankhwala TB "Lomfloks" ayenera pamodzi ndi mankhwala monga "Isoniazid", "pyrazinamide wokhala" ndi "Ethambutol".
Pa nthawi yomweyo ndi osafunika kwambiri kutenga lomefloxacin ndi rifampicin. Ichi ndi chifukwa chakuti zinthu zimenezi ndi mpikisano muzikangana.
Chiopsezo zosiyanasiyana photochemical akhoza kwambiri yafupika potenga Lomfloks mapiritsi ' "madzulo.
Mwanjira mankhwala
Kodi ndingachite mankhwala ena mankhwala "Lomfloks"? Malangizo ntchito (njira ya analogues Adzaperekedwa ku mapeto a nkhani) limanena kuti mankhwala akhoza kuonjezera ntchito anticoagulants m'kamwa, komanso kuonjezera kawopsedwe wa NSAIDs.
Mankhwalawa ayenera kumwedwa ndi sucralfate pang'onopang'ono mayamwidwe mankhwala ndi kuchepetsa bioavailability ake, kupanga pawiri chelate. Pankhani phwando munthawi yomweyo ndi probenecid, izo kumathandiza kuti chopinga wa excretion aimpso.
zotsatira zoyipazi
Kodi kungasokoneze pa thupi mankhwala "Lomfloks"? Malangizo ntchito (ndemanga, analogs m'nkhani ino) limanena kuti ankamuona wothandizila ali zotsatira zotsatirazi mbali:
- Ziwiya ndi mtima: Vasculitis ndi kupondereza ntchito cardio-m'mapapo mwanga dongosolo.
- Kupuma dongosolo: edema a m'mapapo ndi m'phuno.
- Ziwengo: matupi awo sagwirizana zochita, photosensitivity, anaphylaxis ndi angioedema.
- Chimbudzi: pseudomembranous matenda a m'matumbo ndipo soreness wa mucosa m'kamwa.
- Chiwindi: chitukuko cha matenda a chiwindi.
- Mkodzo: polyuria, interstitial nephritis, posungira mkodzo ndi kulephera aimpso.
- Minofu / mafupa: tendonitis, mitsempha chophukacho, arthralgia ndi myalgia.
- Mantha dongosolo (zotumphukira ndi pakati): nkhawa, ataxia, chisokonezo, kupweteka, kuvutika, kenaka utentha mamba, matenda tulo, chizungulire, kusokonezeka maganizo, litsipa, kuyerekezera zinthu m'maganizo, kusawona bwino, mphulupulu kulawa, photophobia ndi diplopia.
- Khungu: hyperpigmentation, exfoliative dermatitis, Stevens-Johnson syndrome ndi epidermal necrolysis.
- Kagayidwe: Hypoglycemia.
- Magazi: haemolytic magazi m'thupi ndi thrombocytopenia.
Kusamala
Yomwe mbali ya mankhwala ayenera kudziwa odwala, asanadye "Lomfloks" piritsi? Kufotokozera lokonzekera, malangizo chofunika kuwerenga, komanso kuyambirira mogwirizana ndi katswiri.
Mu matenda amenewa, monga matenda enaake, ndi kusintha kwa dosing chakudya n'kofunika. Koma izi pokhapokha ngati impso ntchito si akusokoneza.
Pa mankhwala, mankhwala n'kofunika kupewa kukhudzana UV kunyezimira.
Mankhwalawa ayenera kumwedwa, ndi mavitamini, ndi wothandizila ena amene ali zotayidwa, magnesium ndi chitsulo, sayenera kumwedwa maola awiri patsogolo ndi maora awiri kutenga mankhwala pansi kulingalira.
Kodi luso kuyendetsa galimoto ndi kasamalidwe ka mankhwala ndi njira zosiyana, "Lomfloks"? Malangizo ntchito (mtengo wa mankhwala kutchulidwa mu gawo pansipa) imatiuza kuti chida ichi zingachititse chidwi mkhutu ndi chizungulire kwambiri. Pa nkhani imeneyi, n'zotheka ntchito asamagwire ntchito ayenera anaganiza pambuyo poti munthu ziyenera Poyankha wodwalayo kwa mankhwala.
Analogs "Lomfloks" ndemanga mtengo mankhwala
kugwiritsa ntchito ndalama malipoti kalozera waperekedwa m'nkhaniyi (zolinga maphunziro). Monga mtengo, n'zotheka kudziwa mtengo enieni okha pharmacies. Childs, chiwerengerochi zimasiyanasiyana pakati rubles 500 (mapiritsi 5).
Kodi wina kunena za mankhwala "Lomfloks" malangizo ntchito? Analogues wa mankhwala anaitenga mwatsatanetsatane. Malinga ndi iye, mankhwalawa akhoza m'malo ndi mankhwala zotsatirazi: ". Lomefloxacin hydrochloride" "Ksenakvin", "Okatsin", "Lomatsin", "maksakvin", "lomefloxacin", "Lofoks"
Koma ndemanga, iwo ali abwino kwa gawo lalikulu. Odwala kuti "Lomfloks" mapiritsi ndithu bwino kulimbana ndi matenda. Komabe, tisaiwale kuti anthu ena amene mankhwala nthawi zonse kudandaula mavuto.
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