Thanzi, Kukonzekera
"Tolperisone" njira. Malangizo ntchito
Miyala "Tolperisone" zikuphatikizapo gulu la mankhwala, relaxants minofu. The medicament kumakhudza chapakati. Mankhwala ali Kakhungu ofunika ntchito, mitsempha-mopupuluma kubweza atagwira motoneurons ndi yaikulu ulusi afferent. Izi amakwiya Letsani wa poly- ndi monosynaptic bongo msana. Mankhwala kumabwezera mmbuyo ndi conduction wa malemeredwe mu ubongo tsinde njira reticulospinal. Kaya zotsatira za chapakati mantha dongosolo zikutanthauza kuwonjezeka zotumphukira magazi. Kukula amenewa angakhale chifukwa chikoka cha antiadrenergicheskim ndi mankhwala antispasmodic. Kugwiritsa ntchito mankhwala pakamwa zikunenedwa bwino odzipereka kwa intestine yaing'ono. Pambuyo theka la ola, ola pazipita anati ndende pazipita mankhwala plasma. Chifukwa persistemnogo anasonyeza kagayidwe medicament bioavailability 20%. Azingokhala mankhwala akupezeka impso ndi chiwindi. Mu mawonekedwe a metabolites mpaka 99% excreted mu mkodzo.
"Tolperisone" mankhwala. Malangizo ntchito. umboni
Perekani mankhwala pa okwera (pathologically) kamvekedwe ndi kuphipha mu minofu striated kugwirizana ndi kudwala ubongo organic mu zotupa wa kapepalako pyramidal, sitiroko, ofoola ziwalo, encephalomyelitis, kuphatikizapo myelopathy. The medicament "Tolperisone" malangizo Buku akuonetsa mankhwala reductive pambuyo ntchito mu traumatology ndi zamafupa. Mwa zizindikiro ndi monga kuchuluka kamvekedwe ndi minofu kuphipha, akulu contracture, complicating matenda mu dongosolo minofu ndi mafupa. Makamaka mankhwala othandiza mu lumbar ndi ululu khomo lachiberekero syndrome, nyamakazi mu mfundo zikuluzikulu, spondyloarthrosis, spondylosis. Mothandizana ndi njira zina yokonza "Tolperisone 'analimbikitsa malangizo ntchito mankhwala a occlusive mtima mtundu matenda.
"Tolperisone" mankhwala. Malangizo ntchito
mankhwala akutengedwa pa mlingo koyamba wa 50 mg si nthawi zoposa zitatu masana. Pang'onopang'ono kuchuluka kwa anagwira mankhwala kwa 150 mg 2-3 p. / Tsiku. nthawi The anatsimikiza payekha malinga ndi chikhalidwe ndi zovuta boma matenda a wodwalayo.
contraindications
Miyala "tolperisone" (mayankho a akatswiri titsimikizire kuti) ali sanagaŵiridwe makanda pansi zaka 18, tsankho zigawo zikuluzikulu. Contraindications monga mimba ndi mkaka wa m'mawere. Chifukwa kukhalapo kwa lactose mu mankhwala osavomerezeka mankhwala tsankho kapena akusowa wa thunthu.
"Tolperisone" njira. Malangizo ntchito. zosiyanasiyana chokhwima
Mankhwalawa amakwiya mutu, minofu kufooka, nseru, gastralgia (akuthamanga pa mlingo wochepa). Pamaziko a mankhwala limapezeka hypotension, matupi awo sagwirizana anachita chifukwa cha tsankho.
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