Thanzi, Kukonzekera
"Kuyambira": malangizo, mayankho. "Kutsika" (mapiritsi): mtengo
Kodi mumadziwa chiyani za Avodart? Mafotokozedwe, mtengo, zizindikiro ndi malangizo a chida ichi zidzafotokozedwa m'nkhaniyi. Mudzaphunziranso za katundu amene ali nawo mu mankhwala awa, gulu la mankhwala ndi liti, gawo lake, ndi zina zotani.
Fomu, kufotokozera, kupakidwa ndi kupanga
Avodart ya mankhwala imapezeka pamtundu wofewa wa gelatinous oblong ndi opaque capsules a chikasu, otchulidwa ndi code "GX CE2". Pogulitsa mankhwalawa angapezeke m'makatebodi a makatoni, kumene mazira amapezedwa ndi mapiritsi 90 kapena 30.
Dutasideide amagwira ntchito ngati wothandizira, komanso gelatin, butylhydroxytoluene, triglycerides, titanium dioxide, inki yofiira yosindikizira, mono-diglycerides ya caprylic acid, glycerin, lecithin ndi okosijeni ya ferric amagwiritsidwa ntchito monga zowonjezera.
Makhalidwe a Pharmacodynamic
Kodi gulu la mankhwala a Avodart ndi chiyani? Malangizo ogwiritsira ntchito akuti mankhwalawa antiandrogenic. Zomwe zimagwira ntchito ndizomwe zimayambitsa mavitamini a 5-alpha-reductase. Chigawo ichi chimatha kuletsa kutembenuka kwa testosterone ku DHT. Izi zimachokera ku kuchotsedwa kwa ntchito ya 5-alpha-reductase ya mitundu yoyamba ndi yachiwiri.
Pambuyo potenga Avodart, kukodza kumayendera bwino, kukula kwake kwa prostate kumachepa, ndipo mwayi wochiza matenda popanda opaleshoni ukuwonjezeka.
Mbali za mankhwala
Malinga ndi akatswiri, mapiritsi a Avodart amasonyeza mmene mankhwala amathandizira masiku 8-15 atangoyamba kumene. Kuthamanga kwa mlingo wa mankhwalawa, kumakhudza kwambiri kupanga DHT.
Pharmacokinetic katundu
Mankhwalawa "Avodart", omwe mtengo wake umasonyezedwa pansipa, amapezeka m'magazi omwe ali pamwamba pa maola 1.5 maola atalandira. Zowonongeka zake ndi 60%. Kudyako chakudya nthawi imodzi sikungakhudze mbali zamakono za mankhwala.
Wothandizirawa ali ndi mapuloteni a plasma (pafupifupi 99%). Tiyeneranso kukumbukira kuti ndi kudya kwadongosolo komanso kwa nthawi yayitali pafupifupi 12 peresenti ya chogwiritsidwa ntchito chikulowetsa umuna.
Kodi wogwira ntchitoyo amachizidwa bwanji? Kodi malangizo ndi maumboni amati chiyani izi? "Kuthamanga" kumakhala kwakukulu kwambiri mu thupi la munthu. Pafupifupi 2-15% ya mankhwala yogwiritsidwa ntchito amakhala osasinthika kupyolera mu matumbo. Kuchetsa kwa mankhwalawa kumakhala pafupifupi mwezi umodzi kutha kwa maphunzirowo.
Akatswiri amati ngakhale ngakhale patapita miyezi isanu ndi umodzi, mankhwala angapo amapezeka m'magazi.
Zisonyezo
Kodi cholinga cha mankhwalawa n'chiyani? Kodi malangizo ndi ndemanga zimati chiyani za izi? "Kuthamanga" ndi mankhwala omwe amagwiritsidwa ntchito pazifukwa zotsatirazi:
- Ndi monotherapy ndi prophylaxis ya prostatic hyperplasia kupitirira kwa prostate (mawonekedwe abwino) mwa kuchepetsa kukula kwake, kukonzanso kukodza, kuchepetsa zizindikiro, ndi kuchepetsa mwayi wa opaleshoni ndi chiopsezo cha kusungidwa kovuta kwambiri;
- Pogwiritsa ntchito mankhwala omwe ali ndi alpha1-adrenoblockers, komanso kuteteza kupitirira kwa prostatic hyperplasia ya prostate (mawonekedwe oipa) pochepetsa kukula kwake, kuchepetsa kukodza, kuchepetsa zizindikiro, kuchepetsa mwayi wa opaleshoni komanso chiopsezo chokhala ndi ubweya wamakono.
Contraindications
Zaletsedwa kugwiritsa ntchito Avodart pamene:
- Hypersensitivity kwa dutasteride, komanso zinthu zina za mankhwala;
- Kuchulukitsa mphamvu kwa inhibitors ya 5-alpha-reductase.
Tiyeneranso kukumbukira kuti mankhwalawa amavomerezedwa kuti avomereze kwa ana ndi amayi.
Mosamala Avodart ayenera kulamulidwa kuti asakwanira.
Makapulisi apamwamba: malangizo othandizira
Mankhwala amatengedwa pamlomo pokhapokha ngati atadya chakudya.
Ma Capsules amamezedwa kwathunthu, osati kutafuna komanso osatsegulira (zomwe zili mkatizi zingayambitse chipwirikiti cha ntchentche).
Mu BPH, akulu ndi amuna okalamba amapatsidwa mankhwala pa kapu imodzi imodzi kamodzi pa tsiku.
Ngakhale kuti chithandizo cha mankhwalawa chimabwera pakatha masabata awiri, ndibwino kuti mutenge miyezi isanu ndi umodzi.
Avodart angagwiritsidwe ntchito pokhapokha mu monotherapy komanso palimodzi ndi alpha 1-adrenoblockers.
Mankhwala apadera
Pa mlingo wa 500 μg pa tsiku, pafupifupi 0,1% ya mankhwalawa imabisika ndi impso. Pankhani iyi, palibe chifukwa chochepetsera mlingo kwa anthu omwe asokoneza makoswe.
Odwala omwe alibe matenda a chiwindi Avodart ayenera kunyalanyazidwa kwambiri, chifukwa mankhwala ake amayamba kugwiritsidwa ntchito kwambiri m'thupili.
Zovuta zochitika
Ndi zotsatira zotani zomwe zimachitika mukamamwa mankhwalawa? Madokotala amati chiyani izi? Zomwe zingasokoneze zotsatirazi:
- Kusasamala ndi kuvutika maganizo;
- Kuphulika kwa khungu, ming'oma, kutupa, mawonetseredwe opatsirana (mpaka ku angioedema);
- Kutaya tsitsi pamutu pa thupi ndi hypertrichosis;
- Edema wowawa ndi testicular;
- Kuchepetsa libido ndi chilakolako chogonana, kupweteka kwa erectile, kutupa ndi kumva zopweteka za zimbudzi za mammary, mavuto okhwima.
Zomwe zimakhala zovuta kuchitapo kanthu zimachepetsedwa kwambiri ndi kuchuluka kwa mankhwala (mwachitsanzo, kuyambira chaka chachiwiri chotenga capsules).
Ngati mumagwirizanitsa Avodart ndi mankhwala ena, kuchuluka kwa zochitika, komanso zochitika zovuta, zingakhale zosiyana pang'ono.
Malangizo apadera
Ma capsules amtunduwu sangathe kutsegulidwa, komanso kulola kuyanjana ndi zomwe zili mkati mwake ndi mucous membranes ndi khungu zolumikiza. Ngati mankhwalawa akadakali pakhungu, ayenera kutsukidwa nthawi yomweyo ndi madzi.
Kuphatikizidwa kwa dutasteride ndi alpha-adrenoblockers kumawonjezera chiopsezo cha matenda a mtima.
Musanayambe kumwa mankhwala, komanso panthawi ya mankhwalawo, m'pofunika kuti muyambe kufufuza za prostate gland (chiwalo cha rectal, PSA, etc.).
Mtengo wamapirisi ndi zina zotero
Kodi Avodart ndi zochuluka bwanji? Mtengo wa mankhwala awa ndi wapamwamba kwambiri. Mukhoza kugula makapisozi 30 a mankhwalawa kwa 1500-1600 rubles.
Mafananidwe ambiri a Avodart ndi zinthu monga Proscar, Adenosterid, Finpros, Urofin, Prostan, Penester, Finistera.
Mmodzi sangathe kunena kuti mtengo wa mankhwalawa ukhoza kukhala wapamwamba kusiyana ndi makapisozi omwe tikuwaganizira.
Ndemanga
Avodart ndi mankhwala otchuka kwambiri omwe amagwiritsidwa ntchito pochiza ndi kuteteza BPH. Kufufuza za izo kungapezeke kosiyana kwambiri. Odwala ena amanena kuti patatha miyezi 12 kugwiritsa ntchito mankhwalawa prostate gland yachepa kwambiri. Komabe, pakutha kwa chithandizo, icho chinawonjezerekanso. Odwala ena sakondwera kwambiri ndi mtengo wapatali wa mankhwalawa, komanso kuwonongeka kwa erectile komanso kuchepa kwa chilakolako chogonana pamene akulandira.
Akatswiri amanena kuti zochita zoterezi zimatha pokhapokha patatha miyezi 3-4.
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