Thanzi, Kukonzekera
"Felodip": malangizo ntchito, ndemanga. analogues mankhwala
Imene imafuna mankhwala "Felodip"? Malangizo ntchito mankhwala adzakhala anafotokoza m'nkhani m'nkhaniyo. Komanso mwa iwo, inu kuphunzira zimene mankhwala akapatsidwa, kodi mankhwalawo iwo ali, kapena contraindications izi mankhwala, momwe ndalama, amene ali analogues ndi zina zotero.
The zikuchokera mankhwala, mawonekedwe opanga ndi ma CD
Mu mawonekedwe zimene mungazipeze pa mankhwala mankhwala "Felodip"? kugwiritsa ntchito bukuli mankhwala limanena kuti alipo kokha mu mawonekedwe a mapiritsi kanthu yaitali. Komanso Mlingo osiyana mankhwala ali envelopu osiyana:
- mapiritsi chikasu mu mawonekedwe a mphodza, popanda fungo aliyense amaimira chiwerengero 2.5. The yogwira chinthu choterocho mankhwala felodipine amachita zinthu m'njira kuchuluka kwa 2.5 mg. Excipients mankhwala ndi lactose monohydrate, hypromellose, microcrystalline mapadi, okusayidi wofiira chitsulo, povidone, titaniyamu dioxide, propyl gallate, okusayidi chikasu chitsulo, magnesium stearate, propylene glycol, anhydrous colloidal silika, talc. Mu kugulitsa mankhwala yogwira akulowa chithuza miyala 10 kuti anayikidwa mu makatoni.
- Mapiritsi a kuwala pinki mtundu mu mawonekedwe a mphodza, popanda fungo aliyense amaimira chiwerengero 5. The yogwira zikuluzikulu za pochita mutuluka felodipine mu kuchuluka kwa 5 mg. Excipients mankhwala protrude lactose monohydrate, hypromellose, microcrystalline mapadi, okusayidi wofiira chitsulo, povidone, titaniyamu dioxide, propyl gallate, okusayidi chikasu chitsulo, magnesium stearate, propylene glycol, anhydrous colloidal silika, talc. Mu kugulitsa mankhwala yogwira akulowa chithuza miyala 10, anayikidwa mu makatoni.
- Mapiritsi pabuka bulauni mphodza zooneka popanda fungo aliyense anasankha numeral 10. mchitidwe yogwira chotero zochita mankhwala felodipine mu kuchuluka kwa 10 mg. Auxiliaries ndi lactose monohydrate, hypromellose, microcrystalline mapadi, okusayidi wofiira chitsulo, povidone, titaniyamu dioxide, propyl gallate, okusayidi chikasu chitsulo, magnesium stearate, propylene glycol, anhydrous colloidal silika, talc. Mu kugulitsa mankhwala yogwira akulowa chithuza mapiritsi 10. Matuza anaika mu makatoni.
The pharmacological katundu wa mankhwala
ndi chipangizo zachipatala "Felodip" n'chiyani? Malangizo ntchito mankhwala akuti ndi kashiamu njira blocker pang'onopang'ono. Ankaona mankhwala uli gulu la dihydropyridine.
mankhwala akhoza kuchita khama zotsatira antianginal ndi antihypertensive. Komanso kumachepetsa zoipazi (magazi) ndi kucheperachepera zotumphukira mtima kukana.
Kodi katundu wina ndi mankhwala "Felodip"? Malangizo ntchito yokonza kumaphatikizapo mudziwe kuti ali nazo mlingo amadalira odana ischemic kwenikweni. Mankhwala kumachepetsa infarction kukula, komanso amateteza thupi ku matenda reperfusion.
chida ichi ali pafupifupi palibe zoipa inotropic kwenikweni. Iwo ali amadza kochepa dongosolo kuchititsa.
The pharmacokinetics mankhwala
utali mankhwala imatsala, "Felodip"? Malangizo ntchito, ndemanga izi zikutanthauza zimenezo. pambuyo mlingo wa medicament mu mankhwala yogwira pafupifupi atamezedwa kotheratu kwa mundawo m'mimba ndipo amachita nthawi yomweyo. Zikomo kuti maonekedwe ake mlingo anachedwa amasulidwe amafotokozera yogwira zipangitsa ndende ake yunifolomu mu magazi (mkati mwa tsiku), komanso kumabweretsa ndi kuwonjezeka mu gawo mayamwidwe.
Sitingathe kunena kuti bioavailability wa mankhwala sadalira pa mlingo achire ndi pafupifupi 15%.
KUMANGA zonsezo plasma ndi yeniyeni ndi pafupifupi 99%. The medicament adzamasulidwa pamodzi ndi mkaka wa m'mawere ndi likulowerera magazi ubongo chotchinga chotchinga placental. Ndi ntchito yaitali thunthu yogwira palibe kudzikundikira amapezeka.
Kodi mankhwala ndi zimapukusidwa "Felodip"? The yogwira pophika wothandizila izi zimapukusidwa mu chiwindi. Mu mawonekedwe metabolites kulalikira.
Hafu ya moyo wa mankhwala ndi za 25 maola. Anasonyeza kukonzekera monga metabolites (pafupifupi 70%) mu mkodzo ndi ndowe (30%).
zikuonetsa medicament
Nthawi zina, wodwalayo Kwalamulidwa mankhwala "Felodip" (5 mg) Malangizo a mankhwala lili mndandanda wa zikuonetsa ntchito:
- oopsa;
- angina;
- arrhythmia;
- inatsekeratu matenda a mtima;
- matenda magazi;
- Raynaud ndi matenda.
contraindications mankhwala
Imene milandu ndi kutiletsa kumwa mankhwala "Felodip"? Reviews madokotala, komanso malangizo m'munsichi amanena kuti mankhwala ayenera kugwiritsidwa ntchito pa zinthu zotsatirazi:
- pachimake m'mnyewa wamtima infarction, komanso mwa mwezi umodzi pambuyo m'mnyewa wamtima;
- wosakhazikika angina;
- cardiogenic mantha;
- mtima kulephera, makamaka decompensated;
- kung'ambika stenosis (kukomoka kwambiri);
- mimba;
- hypotension (aakulu);
- ana ndi achinyamata (pansi zaka 18);
- pa mkaka wa m'mawere;
- kuchuluka tilinazo wodwalayo mankhwala kapena ofanana nawo ena dihydropyridine.
Mmodzi Tisaiwale kuti chida ichi ndi kusamala kwambiri Kwalamulidwa kwa odwala ndi kwa chiwindi ndi aimpso insufficiency.
Medical chipangizo "Felodip": malangizo ntchito
Analogues chida Adzaperekedwa patsogolo pang'ono. Tsopano ine ndikufuna kuti ndikuuzeni inu za mmene mankhwala ayenera kumwedwa molondola.
Pamene matenda oopsa mlingo akulu ndi anthu okalamba wayikidwa payekha. Childs, kuchuluka koyamba mankhwala ndi 5 mg tsiku lililonse. Pa kusankha odwala yoyenera mlingo akulimbikitsidwa kugwiritsa ntchito piritsi a 2.5 mg. Pamene mwamsanga ayenera kuwonjezera mlingo wa mankhwala akhoza kukhala. Wapakati buku la medicament kwa yokonza mankhwala 5-10 mg wa pa tsiku.
Kwa odwala okalamba kapena odwala ndi opuwala chiwindi ntchito mu mankhwala oyambirira ndi kutumikiridwa mu kuchuluka kwa 2.5 mg wa pa tsiku.
Mankhwala khola angina "Felodip" zotchulidwa payekha. Choncho mlingo koyamba (akuluakulu) ndi 5 mg tsiku lililonse. Ngati chofunika, mlingo akhoza ziwonjezeke kwa mg ndi 10 patsiku. The pazipita tsiku kuchuluka kwa mankhwala ndi 20 mg.
Miyala "Felodip" amaloledwa kutenga osakaniza ndi zoletsa Ace, beta-blockers ndi okodzetsa. Komabe, tisaiwale kuti pamene zotsatira hypotensive kumatheka. Choncho muyenera kusamala kwambiri chifukwa cha chiopsezo hypotension kuchuluka.
Mu odwala kwambiri chakhungu ntchito chiwindi mlingo wa mankhwala ayenera kuchepetsedwa.
Umene mankhwala ayenera kumwedwa m'mawa pamaso kadzutsa. Pankhaniyi, phale Mulimonsemo sikutheka osokoneza, tulo kapena kugawaniza.
njira ambiri osokoneza
ntchito pachithunzichi mapilisi "Felodip" zizindikiro zotsatirazi cha mankhwala osokoneza bongo kumachitika odwala: bradycardia ndi hypotension (aakulu).
Mu nkhani ya yatsoka zizindikiro ngati symptomatic mankhwala. Ngati hypotension (aakulu) odwala kupereka malo yopingasa ndi kukweza miyendo. Mokhudzana bradycardia, mu nkhani imene atropine mtima intramuscularly kutumikiridwa pa mlingo wa 0.5-1 mg. Ngati ndi kotheka, kuonjezera buku la madzi kulowetsedwa ikuchitika ndi sodium kolorayidi, shuga njira kapena dextran.
Pamene pamwambapa anafotokoza inefficiency miyeso Kwalamulidwa mankhwala wodwala ndi zotsatira osakhala pa zolandilira alpha-adrenergic.
Zotsatira zake zoyipa ku kutenga mankhwala
Kodi kungasokoneze thupi kumwa mankhwalawa "Felodip"? Analogues chida ndi kukonzekera pakokha amachititsa mutu, ankatenthetsa nkhope, chizungulire, palpitations ndi kutopa. Komabe, tisaiwale kuti maganizo ndi kusintha. Iwo kawirikawiri amaoneka pa chiyambi cha mankhwala, komanso ndi kuwonjezeka mlingo wa mankhwala.
Mwa njira, malingana ndi kuchuluka analandira mankhwala wodwala angaoneke ndi edema zotumphukira. Malinga ndi akatswiri, iwo amakhala vasodilation precapillary.
Odwala ndi periodontal kapena chiseyeye odwala kulandira mankhwala akhoza kukhala chotupa ka usinini. Zimenezi zikhoza kupewedwa ngati inu kusunga mokwanira m'kamwa ukhondo.
Nthawi zina timakhala tikulingalira kulandira mankhwala amakhala chifukwa cha zotsatira otsatirawa mbali:
- dongosolo mtima: palpitations, tachycardia, ndi edema zotumphukira.
- zochita Dermatological: photosensitivity, pruritus, urticaria.
- Zotumphukira ndi chapakati mantha dongosolo: paresthesia, kupweteka chizungulire.
- dongosolo minofu ndi mafupa: arthralgia, myalgia.
- M'mimba thirakiti: gingival hyperplasia, nseru, kuwonjezeka mu michere chiwindi.
- Other: kutopa, zochita hypersensitivity, kuphatikizapo angioedema.
Analogs, ndipo mtengo wa mankhwala
Kodi ndindalama mankhwala pamaso pathu? Kuti ndi nkhani anakweza ndi odwala ambiri kulandira mankhwala ino kutumikiridwa. Tikumbukenso kuti lero ndi mankhwala zikhoza kugulidwa pa mitengo zotsatirazi:
- Mapiritsi a 2.5 mg (zidutswa 30) - 425 Russian rubles;
- mapiritsi mu buku la 5 mg (zidutswa 30) - 556 Russian rubles;
- mapilitsi mu buku la mg wa 10 (zidutswa 30) - 831 Russian rubles.
Kodi m'malo mankhwala "Felodip"? Analogs za mankhwala akupezeka pafupifupi aliyense mankhwala. Pakati pawo, ine ndikufuna kuti asonyeze mankhwala zotsatirazi:. "Plendil," "Felodipine-NW", "Felodipine" ndi "Felotenz achigonjetse"
Zabwino mayankho ochokera odwala za mankhwala mankhwala
Umboni za "Felodip" kukonzekera boma kuti kwambiri ogwira ndi bwino analekerera ndi odwala, mosasamala kanthu za msinkhu komanso jenda. Komanso, yogwira mankhwala akhoza kumwedwa ngakhale odwala matenda a shuga, matenda aimpso, mphumu komanso nthenda zina obstructive m'mapapo ndi matenda Raynaud a, hyperlipidemia, gout, ndipo pambuyo m'mapapo kupatsidwa zina.
Akatswiri ambiri amanena chakuti mankhwala alibe zotsatira pa zamadzimadzi mbiri ndi shuga magazi ndende.
ndemanga zoipa
Pakati pa ndemanga zoipa zimene kusiya odwala pa mankhwala, tingathe kuona kuti anthu zokhudzana ndi kukwera mtengo kwa mankhwala. Ngakhale mankhwala amanena kuti mtengo wake ndi mtima wonse mogwirizana ndi dzuwa ndi khalidwe.
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