Thanzi, Kukonzekera
"Flyuanksol": malangizo ntchito, madokotala weniweni. Zotsatira zoyipa "Flyuanksola" analogues wa mankhwala
ndi mankhwala "Flyuanksol" n'chiyani? Malangizo ntchito mankhwala, zosakaniza ake, zotsatira zoyipazi, mawonekedwe kumasuka ndi katundu pharmacological zafotokozedwa mwatsatanetsatane m'nkhani ino. Kuyambira mungathe kuphunzira zimene contraindications ndi zizindikiro wanena mankhwala, momwe ndalama, zimene zidzachitike mu nkhani ya mankhwala osokoneza bongo, ndi zina zotero D..
The zikuchokera mankhwala ndi kutulutsidwa zikuluzikulu
Kodi mfundo yogwira lili mankhwala "Flyuanksol"? malangizo ntchito za malangizo medicament limanena kuti ngati chigawo yogwira izo mutuluka hydrochloride flupenthixol.
Monga mawonekedwe a kumasulidwa, koma lero ndi njira lingapezeke mu madontho, miyala ndi njira, ndi mafuta ofotokoza anafuna makonzedwe mu mnofu. Mankhwala woyamba akugulitsa galasi zatemennom 10 ml, chachiwiri - mu katoni 100 kapena 50 ndi wachitatu - mu ampoules zidutswa 10.
General katundu wa mankhwala
N'chifukwa chiyani mankhwala "Flyuanksol"? Umboni za mankhwala omwe anapereka m'munsimu. Mapiritsi ndi jekeseni ndi gulu la antipsychotics. Iwo adzalandira anxiolytic, antidepressant ndi zotsatira sedative. Zabwino ndemanga za mankhwala zili ndi mfundo zimene mosabvuta imayendetsa boma maganizo a wodwalayo komanso kumathandiza kuti anatengera chikhalidwe.
Makhalidwe pharmacological mankhwala
ndi makhalidwe a pharmacological mankhwala "Flyuanksol" n'chiyani? Malangizo ntchito akusonyeza kuti mankhwala ndi neuroleptic kutchinga zolandilira adrenergic ndi maselo dopamine mu ubongo. Chifukwa cha chinthu yogwira zimatheka sedation. Childs, izi zimachitika pa 8-day mlingo zonse.
Kodi odwala za mankhwala "Flyuanksol"? Reviews odwala muli zambiri zosangalatsa. Nthawi zambiri, iwo dziwani kuti mankhwala m'malo mofulumira kumatha zizindikiro za psychosis ndi maganizo, komanso kumathandiza kuti kubwezeretsa maganizo. Odwala matenda sakonda, ndi sociable kusintha kwa anthu.
Features mankhwala
Kodi mankhwala "Flyuanksol"? Reviews madokotala ndi akatswiri ena amanena kuti mbali za mankhwala ndi kuti, malingana ndi mlingo akhoza kuchita wodwala m'njira zosiyanasiyana.
zotsatira Antipsychotic kuwawonetsera pambuyo ntchito medicament zikutanthauza mu kuchuluka kwa 3 mg wa pa tsiku. Mwa njira, mphamvu ya mmene kumawonjezera ndi mlingo.
Kuchuluka kwa 25 mg pa tsiku mankhwala ziribe mphamvu sedative. Komabe, tisaiwale kuti pa mlingo waukulu, zikhoza kuyambitsa zotsatira si yeniyeni sedative.
Pa mlingo osiyanasiyana anasankha wothandizila neuroleptic ali ndi kutchulidwa anxiolytic kwenikweni. Ntchito mlingo ang'onoang'ono (mpaka pafupifupi 3 mg wa pa tsiku), mankhwala ingakhale monga mankhwala ochiritsira antidepressant.
Choncho, mankhwala "Flyuanksol" akhoza kuchepetsa zizindikiro zazikulu za psychosis, kuphatikizapo zinyengo akhate, kuyerekezera zinthu m'maganizo ndi ndinaganiza matenda. Iwo ali katundu disinhibitory (i.e. activating ndi antiautisticheskim) ndipo kumachepetsa ndi maganizo, zomwe pamapeto pake amalimbikitsa kutsegula odwala ndi zizindikiro maganizo anatengera anzawo facilitates ndipo umatithandiza asamangochita zimene akufuna.
Zambiri za mtundu injectable
Kukonzekera "Flyuanksol Depot" ndi njira mafuta anafuna jekeseni mu mnofu zofikira. M'mawu ena, mankhwala uyikidwa mawonekedwe flupenthixol.
Pamene ntchito njira imeneyi pa mlingo ang'ono ndi sing'anga (mpaka 100 mg lililonse masiku 14) kuti wodwalayo si unspecific sedation. Ngakhale akadali kukula pa mlingo waukulu.
Kodi akatswiri amanena za mtundu uwu wa mankhwala ( "Flyuanksol Depot")? Reviews kupereka zimenezi Njira wautali nthawi yopeza wodwalayo, osati miyala mankhwala. Komanso, kuthokoza kwa iye, n'zosavuta kuchita mosalekeza antipsychotic chithandizo, umene uli wofunika kwambiri kwa odwala amene Musatenge kunja mankhwala kuchipatala.
Kuchokera pamwamba Ndizachidziwikire kuti mankhwala "Flyuanksol Depot" ndi kuteteza musabise kawirikawiri kugwirizana ndi mowiriza kusokoneza mankhwala. Mu mnofu jekeseni angathe kuchitidwa pa intervals wa masabata awiri kapena anayi.
Pharmacokinetics
Kodi mwakhala nthawi yotani odzipereka mankhwala "Flyuanksol"? Pambuyo makonzedwe m'kamwa ndende pazipita amafotokozera yogwira zimatheka pafupifupi 3-7 maola madzi. The bioavailability wa mankhwala ndi 40%.
Yogwira chinthu mankhwala pang'ono likulowerera chotchinga placental. Iwo ayenera kukumbukira kuti, zochepa, izo yafotokozedwa ndi mkaka wam'mawere. Zodabwitsa ndizakuti, ndi metabolites ndi ntchito neuroleptic.
Kodi jekeseni "Flyuanksol Depot"? Guide limanena kuti pambuyo mu mnofu jekeseni wa mankhwala CIS (Z) -flupentixol decanoate amaloŵamo pogawanikana pamawere (enzymatic). Izi ndipamene zinthu yogwira wa CIS (Z) -flupentixol acid decanoic. Ndende abwere ku seramu zimatheka choyamba cha kumapeto kwa sabata loyamba pambuyo jekeseni.
Pamene kulandira miyala mu nyengo awo kuswana 35 maola. Ngati panali ntchito njira jekeseni, ndende amachepetsa exponentially mu seramu (pambuyo masabata 3).
Anasonyeza yogwira medicament mu mawonekedwe a metabolites kudzera intestine, ndi impso.
Zikuonetsa ntchito wothandizila neuroleptic
Nthawi zina, mankhwala chimasonyeza "Flyuanksol"? Zimenezi zikhoza kukhala zosiyana, malingana ndi mlingo.
mankhwala imaonekera pa mlingo mpaka 3 mg wa pa tsiku zotsatirazi zinthu pathological:
- maganizo wofatsa ndi digiri zolimbitsa, limodzi ndi kutopa, nkhawa komanso kusowa kanthu;
- matenda choganiza kuti kumawonetsera ndi zochita asthenic;
- matenda neurotic (aakulu), limodzi ndi mphwayi, maganizo ndi nkhawa;
- ndi pachimake situational nkhawa matenda, komanso chikhalidwe cha maganizo kwambiri maganizo, musati amafuna sedative kapena zotsatira zachinyengo (mwachitsanzo, ngati wodwala kumwa asamakhale ndi nkhawa).
Medicament "Flyuanksol", analogues limene Adzaperekedwa kumapeto kwa nkhani, anamusankha pa Mlingo wa 3 mg wa pa tsiku ndipo ngati pali kupatuka zotsatirazi: zinthu psychotic amene anatsagana ndi zinyengo akhate, kuyerekezera zinthu m'maganizo, chisokonezo maganizo, anergy, mphwayi ndipo satha kulankhula bwinobwino.
Contraindications ntchito wothandizila neuroleptic
Mu zina, ali osavomerezeka ntchito mankhwala "Flyuanksol"? Malangizo ntchito monga mndandanda kutsatira contraindications:
- zaka ana (zaka 18);
- CNS maganizo;
- mkaka wa m'mawere;
- pa mimba;
- Kuledzela (pachimake) barbiturates;
- kusokonekera;
- Kuledzela pachimake opioid analgesics;
- pheochromocytoma;
- mowa pachimake poyizoni;
- comatose limati;
- mafupa yimitsira;
- kusintha pathological m'mwazi;
- hypersensitivity kuti neuroleptics ndi dongosolo tioksantenoviy.
Iwo ayenera kukumbukira kuti si bwino kuti mankhwala mankhwala pa mlingo yaing'ono (3 mg) mu mkhalidwe ofuntha kapena excitations.
Mankhwala "Flyuanksol": malangizo (mapiritsi, ukutsika)
Zochizira nkhawa ndi maganizo matenda mlingo woyambilira wa medicament a mapiritsi ayenera 1 mg tsiku lililonse (makamaka m'mawa), kapena 500 mcg kawiri pa tsiku. Ngati zotsatira achire palibe, kuchuluka kwa mankhwala sabata akhoza ziwonjezeke kwa 2 mg. Choncho mlingo tsiku (2-3 mg) kugawidwa mu magawo angapo. Ngati mmene palibe pamene ntchito mankhwala mlingo yayikulu (i.e., 3 mg), ndiye ayenera kuchotsedwa.
Mankhwalawa zinthu psychotic anapereka kuchuluka kwa mankhwala payekha yekha. Koyamba tsiku mlingo akhale 3-15 mg wa pa mlingo 3 anagawa. Ngati n'koyenera, buku anati akhoza ziwonjezeke kwa mg ndi 20 kapena 30 patsiku. Mlingo pazipita sayenera oposa 40 mg.
Monga ankaimira wothandizila yokonza mankhwala ndi kutumikiridwa mu kuchuluka kwa 5-20 mg ndi kamodzi patsiku (m'mawa).
Koma dontho "Flyuanksol", iwo ayenera kumwedwa mkati. Madokotala zambiri mankhwala mankhwala ofunikira okha ngati pazifukwa zosiyanasiyana, simungathe kutenga mankhwala pakamwa (piritsi). Wothandiza mlingo odwala ndi 4-40 mg wa pa tsiku.
Jekeseni "Flyuanksol": malangizo, ndemanga mtima
Yankho wochuluka kwa jekeseni mu mnofu zofikira ayenera kuperekedwa yozama nusu chapamwamba kunja kwa matako a. Mlingo ndi imeneyi pakati mankhwala ayenera kuikidwa payekha (palokha mmene achire).
chiphunzitso ichi kawirikawiri ntchito mu kuchuluka kwa 20-40 mg (kapena 1-2 ml) pa masabata 2 kapena 4. Tikumbukenso odwala ena kungafune Mlingo zazikulu ndi lalifupi imeneyi pakati jekeseni.
Ngati anasankha buku la mankhwala a jekeseni (20 mg / ml) ndi oposa 2 kapena 3 ml ya 1 ndondomeko, m'pofunika kuyenda ndi njira ya ndende mkulu.
Kukonzekera 100 mg / ml ya ayenera kubayidwa mu buku la 50-200 mg (kapena 0.5-2 ml) pa masabata 2-4. Mu muyambirenso pachimake kapena exacerbation la matenda zina zimafunika kamodzi oyamba akutanthauza ndalama mpaka 400 mg pa intervals a 2 kapena 1 sabata. Pambuyo zizindikiro pachimake pochitika, inu anfunika kubala kuchepetsa pang'onopang'ono mlingo kwa yokonza ndi (20-200 mg wa pa masabata 2-4).
Ngati chofunika yakubuluka mawonekedwe m'kamwa wa mankhwala kwa parenteral kukonzekera wothandiza mankhwala Ndi bwino kukhala ndi maziko chiwembu zotsatirazi:
- tsiku kuchuluka (mu mg) wa mankhwala a mapiritsi × 4 = mlingo umodzi (mu mg) jekeseni aliyense masiku 14.
Iwo ayenera kukumbukira kuti mkati mwa sabata imodzi pambuyo utsogoleli wa mankhwala akulangizidwa kupitirizabe mankhwala a mapiritsi, koma pa mlingo m'munsi. Yotsatira voliyumu ndi kusiyana pakati pa njira anakhazikitsa malinga ndi zotsatira achire.
Zolemba malire mlingo injectable njira (wina gawo) ndi 400 mg. Choncho kusiyana jakisoni ayenera kukhala pa sabata.
Malinga ndi mayankho odwala, pamene tigwiritsa ntchito bwino kukonzekera ndi kusunga malangizo kuchipatala, ali ndi ubwino mkhalidwe wawo wonse maganizo.
zotsatira zoyipazi
Kodi zoyipa pa thupi mankhwala "Flyuanksol"? Zotsatira zake zoyipa alipo mu mankhwala, kaya mawonekedwe ake. Apa tsopano.
- mantha dongosolo: giperkinetiko-hypertensive matenda (extrapyramidal kuunika), kufooka, akathisia, kufooka, chizungulire, psychomotor retardation, tardive dyskinesia, zochita dystonic ndi neuroleptic matenda oopsa.
- Mtima ndi magazi zotengera: tachycardia, hypotension, orthostatic.
- dongosolo hematopoietic: granulocytopenia.
- Zinthu ziwalo: chosokoneza wa malawi.
- GI: kudzimbidwa, matenda a chikasu ndiyo cholestatic, pakamwa youma, kusintha chosakhalitsa mu mayesero ntchito chiwindi.
- Endocrine dongosolo: kunenepa, galactorrhea, thukuta, gynaecomastia, kusabala, dysmenorrhea, kuchuluka njala, kuchepa libido, azimva kutentha.
- dongosolo mkodzo: mkodzo posungira.
- Chifuwa: dermatitis, photosensitivity, ndi ziwengo.
malangizo Special ntchito
Ndi kwambiri kusamala mankhwala Kwalamulidwa kwa odwala matenda a mtima, matenda convulsive, kulephera kupuma, khungu, matenda Parkinson, zilonda zam'mimba ndi m'matumbo 12 tiperstnoj, mphumu, uchidakwa, ndiko kumayambitsa posungira mkodzo, kulephera chiwindi, ndi otchedwa benign prostatic hyperplasia.
Ngati wodwala ali kale analandira neuroleptics kapena tranquillizers ndi zotsatira sedative, m'pofunika kusiya kumwa iwo bwino.
Pamene yaitali mankhwala, makamaka pa Mlingo mkulu analimbikitsa kulamulira ndi kuunikira mmene alili pofuna kukonza yokonza mlingo.
Mankhwalawa munthawi yomweyo shuga ntchito anati chiphunzitso kungafune kudzudzulidwa kuchuluka kwa insulin.
Mu ntchito neuroleptics angathe neuroleptic zilonda matenda. zizindikiro zake zazikulu ndi minofu chinthu chimodzimodzi, hyperthermia, asintha udindo maganizo, ndi kukanika wa mantha dongosolo autonomic. Zizindikiro amenewa amafuna mwamsanga Kulipira poika mankhwala ndi wothandiza symptomatic mankhwala.
Nthawi zambiri mankhwala "Flyuanksol" sayambitsa sedation. Koma, ngakhale, m'pofunika kuganizira mmene iye ikhudzire luso bwinobwino ntchito makina, kapena njira zina. Ndikufuna kuona kuti pa mankhwala (makamaka poyamba), odwala ayenera kupewa ntchito zingakhale woopsawo (kudziwa poyankha mankhwala).
Nthawi cha mankhwala osokoneza bongo
Ngati mankhwala amatengedwa bwino (kukweza), izo zingachitike ambiri osokoneza. Pankhaniyi, akusonyeza makhalidwe zotsatirazi: hypo- kapena hyperthermia, kugona, khunyu, matenda extrapyramidal, mantha, hypotension ndi chikomokere.
Kodi kuchita zimenezo? M'pofunika kuchita lothandizana ndi symptomatic mankhwala. Ngati mankhwala anali ingested, kufunika mofulumira kusamba kunja m'mimba, komanso kutenga sorbent. Komanso, n'kofunika kwambiri kuthandiza ntchito za ziwiya, mtima ndi njira kupuma. Iwo ali osavomerezeka ntchito Epinephrine monga kungayambitse kuchepetsa magazi. Zizindikiro Extrapyramidal n'zotheka kusiya mankhwala "Biperiden" ndi khunyu - "ntchito diazepam".
Mogwirizana ndi mankhwala ena
Pamene pogwiritsa ntchito gawo la anati medicament akhoza nakweza zotsatira sedative wa barbiturates, Mowa, ndi wothandizila ena amene zotsatira ochepetsera pa CNS.
Kukonzekera "Flyuanksol kuti" osavomerezeka ntchito molumikizana ndi guanethidine ndi mankhwala Mankhwala ndi zotsatira ofanana. Chimenechi ndi chifukwa chakuti antipsychotics akhoza ndithu wofooka zotsatira zawo antihypertensive.
Ndi limodzi ntchito medicament "Flyuanksol" akhoza kuchepetsa efficacy wa mankhwala "levodopa" ndipo atumiki ena adrenergic.
Pa nthawi yomweyo kutenga mankhwala ndi "Piperazine" ndi "MCP" kwambiri kumaonjezera ngozi ya matenda extrapyramidal.
Iwo ayenera kukumbukira kuti mankhwala neuroleptic kuperekedwa monga njira jekeseni Mulimonsemo sayenera wothira madzi ena.
Price ndi analogues wa mankhwala
Kodi zambiri ndi mankhwala "Flyuanksol"? mtengo wake si mkulu. Choncho, chifukwa mapiritsi 50 1 mg wa inu kulipira pafupifupi 500 Russian rubles. Ngati mukufuna 100 5 mg, iwo zikhoza kugulidwa kwa 1,200 rubles. Koma mawonekedwe jekeseni wa mankhwala, ndiye mtengo kwambiri. Pa 10 Mbale (20 mg / ml) mankhwala amafuna za 2300 rubles.
Kodi ngati wodwalayo sangathe kugula mankhwala "Flyuanksol"? analogues ake amagulitsidwa pafupifupi onse maunyolo mankhwala. Ena mwa iwo ndi izi:
- The njira "Flyuanksol Depot". Ndi mofulumira ndi wamphamvu kwambiri mankhwala. Komabe, miyala kwambiri zodula.
- "Klopiksol" mankhwala. Mtengo uli pafupi kwambiri ku chiyambi. Iwo umapita pa malonda a mapiritsi ndipo ali ndi contraindications ochepa.
- "Truksal" njira. Anagulitsa mapiritsi. The mwayi waukulu mokomera ntchito ana ndi 3-zaka. Ndalama pang'ono pamwamba wapachiyambi.
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